The asymmetric synthesis of β-haloaryl-β-amino acid derivatives

S. D. Bull, S. G. Davies*, S. Delgado-Ballester, G. Fenton, P. M. Kelly, A. D. Smith

*Corresponding author for this work

Research output: Contribution to journalArticlepeer-review

83 Citations (Scopus)

Abstract

Lithium N-benzyl-N-α-methyl-4-methoxybenzylamide is employed as a homochiral ammonia equivalent for the asymmetric synthesis of β-haloaryl-β-amino acid derivatives using a conjugate addition/oxidative deprotection strategy.

Original languageEnglish
Pages (from-to)1257-1260
Number of pages4
JournalSynlett
Issue number9
Publication statusPublished - 1 Jan 2000

Keywords

  • β-haloaryl β-amino acids
  • Asymmetric synthesis
  • Homochiral ammonia equivalent
  • Oxidative debenzylation

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