The asymmetric synthesis of β-haloaryl-β-amino acid derivatives

S. D. Bull; S. G. Davies; S. Delgado-Ballester; G. Fenton; P. M. Kelly; A. D. Smith

The asymmetric synthesis of β-haloaryl-β-amino acid derivatives

S. D. Bull, S. G. Davies^*, S. Delgado-Ballester, G. Fenton, P. M. Kelly, A. D. Smith

^*Corresponding author for this work

Research output: Contribution to journal › Article › peer-review

Abstract

Lithium N-benzyl-N-α-methyl-4-methoxybenzylamide is employed as a homochiral ammonia equivalent for the asymmetric synthesis of β-haloaryl-β-amino acid derivatives using a conjugate addition/oxidative deprotection strategy.

Original language	English
Pages (from-to)	1257-1260
Number of pages	4
Journal	Synlett
Issue number	9
Publication status	Published - 1 Jan 2000

Keywords

β-haloaryl β-amino acids
Asymmetric synthesis
Homochiral ammonia equivalent
Oxidative debenzylation

Cite this

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title = "The asymmetric synthesis of β-haloaryl-β-amino acid derivatives",

abstract = "Lithium N-benzyl-N-α-methyl-4-methoxybenzylamide is employed as a homochiral ammonia equivalent for the asymmetric synthesis of β-haloaryl-β-amino acid derivatives using a conjugate addition/oxidative deprotection strategy.",

keywords = "β-haloaryl β-amino acids, Asymmetric synthesis, Homochiral ammonia equivalent, Oxidative debenzylation",

author = "Bull, {S. D.} and Davies, {S. G.} and S. Delgado-Ballester and G. Fenton and Kelly, {P. M.} and Smith, {A. D.}",

year = "2000",

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language = "English",

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journal = "Synlett",

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T1 - The asymmetric synthesis of β-haloaryl-β-amino acid derivatives

AU - Bull, S. D.

AU - Davies, S. G.

AU - Delgado-Ballester, S.

AU - Fenton, G.

AU - Kelly, P. M.

AU - Smith, A. D.

PY - 2000/1/1

Y1 - 2000/1/1

N2 - Lithium N-benzyl-N-α-methyl-4-methoxybenzylamide is employed as a homochiral ammonia equivalent for the asymmetric synthesis of β-haloaryl-β-amino acid derivatives using a conjugate addition/oxidative deprotection strategy.

AB - Lithium N-benzyl-N-α-methyl-4-methoxybenzylamide is employed as a homochiral ammonia equivalent for the asymmetric synthesis of β-haloaryl-β-amino acid derivatives using a conjugate addition/oxidative deprotection strategy.

KW - β-haloaryl β-amino acids

KW - Asymmetric synthesis

KW - Homochiral ammonia equivalent

KW - Oxidative debenzylation

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M3 - Article

AN - SCOPUS:0033804490

SN - 0936-5214

SP - 1257

EP - 1260

JO - Synlett

JF - Synlett

IS - 9

ER -

The asymmetric synthesis of β-haloaryl-β-amino acid derivatives

Abstract

Keywords

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