Electrophilic fluorination in the synthesis of new fluoroindoles

H F  HODSON; D J  MADGE; Alexandra Martha Zoya Slawin; D A  WIDDOWSON; D J  WILLIAMS

doi:10.1016/S0040-4020(01)80862-0

Electrophilic fluorination in the synthesis of new fluoroindoles

H F HODSON, D J MADGE, Alexandra Martha Zoya Slawin, D A WIDDOWSON, D J WILLIAMS

Research output: Contribution to journal › Article › peer-review

Abstract

Fluorination of trialkylstannylindoles with caesium fluoroxysulfate or Selectfluor(TM) was investigated for the synthesis of inter-alia 2- and 3-fluoroindoles. Caseium fluoroxysulfate gave good yields of these potentially useful intermediates; Selectfluor provided lower yields.

Original language	English
Pages (from-to)	1899-1906
Number of pages	8
Journal	Tetrahedron
Volume	50
Issue number	6
DOIs	https://doi.org/10.1016/S0040-4020(01)80862-0
Publication status	Published - 7 Feb 1994

Keywords

CESIUM FLUOROXYSULFATE
INDOLES

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10.1016/S0040-4020(01)80862-0

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title = "Electrophilic fluorination in the synthesis of new fluoroindoles",

abstract = "Fluorination of trialkylstannylindoles with caesium fluoroxysulfate or Selectfluor(TM) was investigated for the synthesis of inter-alia 2- and 3-fluoroindoles. Caseium fluoroxysulfate gave good yields of these potentially useful intermediates; Selectfluor provided lower yields.",

keywords = "CESIUM FLUOROXYSULFATE, INDOLES",

author = "HODSON, {H F} and MADGE, {D J} and Slawin, {Alexandra Martha Zoya} and WIDDOWSON, {D A} and WILLIAMS, {D J}",

year = "1994",

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T1 - Electrophilic fluorination in the synthesis of new fluoroindoles

AU - HODSON, H F

AU - MADGE, D J

AU - Slawin, Alexandra Martha Zoya

AU - WIDDOWSON, D A

AU - WILLIAMS, D J

PY - 1994/2/7

Y1 - 1994/2/7

N2 - Fluorination of trialkylstannylindoles with caesium fluoroxysulfate or Selectfluor(TM) was investigated for the synthesis of inter-alia 2- and 3-fluoroindoles. Caseium fluoroxysulfate gave good yields of these potentially useful intermediates; Selectfluor provided lower yields.

AB - Fluorination of trialkylstannylindoles with caesium fluoroxysulfate or Selectfluor(TM) was investigated for the synthesis of inter-alia 2- and 3-fluoroindoles. Caseium fluoroxysulfate gave good yields of these potentially useful intermediates; Selectfluor provided lower yields.

KW - CESIUM FLUOROXYSULFATE

KW - INDOLES

U2 - 10.1016/S0040-4020(01)80862-0

DO - 10.1016/S0040-4020(01)80862-0

M3 - Article

SN - 0040-4020

VL - 50

SP - 1899

EP - 1906

JO - Tetrahedron

JF - Tetrahedron

IS - 6

ER -

Electrophilic fluorination in the synthesis of new fluoroindoles

Abstract

Keywords

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