Research output per year
Research output per year
Research output
- 5 Article
Search results
-
2023
Alzheimer’s disease-like neuropathology in three species of oceanic dolphin
Vacher, M. C., Durrant, C. S., Rose, J., Hall, A. J., Spires-Jones, T. L., Gunn-Moore, F. & Dagleish, M. P., 1 Apr 2023, In: European Journal of Neuroscience. 57, 7, p. 1161-1179 19 p.Research output: Contribution to journal › Article › peer-review
Open AccessFile -
Development of submicromolar 17β-HSD10 inhibitors and their in vitro and in vivo evaluation
Benek, O., Vaskova, M., Miskerikova, M., Schmidt, M., Andrys, R., Rotterova, A., Skarka, A., Hatlapatkova, J., Karasova, J. Z., Medvecky, M., Hroch, L., Vinklarova, L., Fisar, Z., Hroudova, J., Handl, J., Capek, J., Rousar, T., Kobrlova, T., Dolezal, R. & Soukup, O. & 3 others, , 5 Oct 2023, In: European Journal Of Medicinal Chemistry. 258, 18 p., 115593.Research output: Contribution to journal › Article › peer-review
Open AccessFile -
2018
1-(Benzo[d]thiazol-2-yl)-3-phenylureas as dual inhibitors of casein kinase 1 and ABAD enzymes for treatment of neurodegenerative disorders
Benek, O., Hroch, L., Aitken, L., Gunn-Moore, F., Vinklarova, L., Kuca, K., Perez, D. I., Perez, C., Martinez, A., Fisar, Z. & Musilek, K., 2018, In: Journal of Enzyme Inhibition and Medicinal Chemistry. 33, 1, p. 665-670 6 p.Research output: Contribution to journal › Article › peer-review
Open AccessFile -
2017
6-benzothiazolyl ureas, thioureas and guanidines are potent inhibitors of ABAD/17β-HSD10 and potential drugs for Alzheimer's disease treatment: design, synthesis and in vitro evaluation
Benek, O., Hroch, L., Aitken, L., Dolezal, R., Guest, P., Benkova, M., Soukup, O., Musil, K., Hughes, R., Kuca, K., Smith, T. K., Gunn-Moore, F. & Musilek, K., Jun 2017, In: Medicinal Chemistry. 13, 4, p. 345-358 14 p.Research output: Contribution to journal › Article › peer-review
Open AccessFile -
In vitro assay development and HTS of small molecule human ABAD/17β-HSD10 inhibitors as therapeutics in Alzheimer’s Disease
Aitken, L., Baillie, G., Pannifer, A., Morrison, A., Jones, P. S., Smith, T. K., McElroy, S. P. & Gunn-Moore, F. J., Jul 2017, In: SLAS Discovery. 22, 6, p. 676-685 11 p.Research output: Contribution to journal › Article › peer-review
Open AccessFile